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首页- Products - Metabolic Enzyme/Protease - Dehydrogenase - AGI-5198

AGI-5198

CAS No. 1355326-35-0

AGI-5198 ( (IDH-C35) )

产品货号. M11453 CAS No. 1355326-35-0

AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.

纯度: >98%(HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
5MG	￥259	有现货
10MG	￥421	有现货
50MG	￥624	有现货
100MG	￥1021	有现货
200MG	获取报价	有现货
500MG	获取报价	有现货
1G	获取报价	有现货

拼团产品询价大包装询价加入购物车

生物学信息

产品名称

AGI-5198
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.
产品描述

AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.
同义词

(IDH-C35)
通路

Metabolic Enzyme/Protease
靶点

Dehydrogenase
受体

R132C-IDH1; R132H-IDH1
研究领域

Cancer
适应症

——

化学信息

CAS Number

1355326-35-0
分子量

462.57
分子式

C27H31FN4O2
纯度

>98%(HPLC)
溶解度

Ethanol: 14 mg/mL (30.26 mM); DMSO: 24 mg/mL (51.88 mM)
SMILES

O=C(NC1CCCCC1)C(N(C2=CC=CC(F)=C2)C(CN3C=CN=C3C)=O)C4=CC=CC=C4C
化学全称

N-cyclohexyl-2-(N-(3-fluorophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido)-2-(o-tolyl)acetamide

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1.Rohle D, et al. Science, 2013, 340(6132), 626-630.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

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